Articaine: uses, dosing, side effects & brands
Articaine is a medicine sold in the U.S. under one brand. Below: what the FDA label says, every product that contains it, what the pills look like, and its recall record.
Key facts
- Available as
- Drops
- Sold as
- Cyklx
- Prescription?
- Prescription only
- Generic available?
- Not in our catalog
Every articaine product we track (1)
Same active ingredient — different manufacturer, form, price and FDA recall record. That last one is what our independent score measures.
Only one: Cyklx.
Combination products containing articaine
A combination is a different drug — different dosing, different warnings. It is listed here so you can find it, not so you can substitute it.
Articaine and breastfeeding
From LactMed, the US National Library of Medicine’s Drugs and Lactation Database — quoted, not rewritten.
Full LactMed record for articaine: levels in milk, effects in breastfed infants, and the drugs it would consider insteadBased on the low excretion of articaine into breastmilk, a single dose of articaine injected during breastfeeding is unlikely to adversely affect the breastfed infant.
National Institute of Child Health and Human Development, record revised June 15, 2025. LactMed states its information is not a substitute for professional judgement.
What people report to the FDA about articaine
The FDA Adverse Event Reporting System (FAERS) collects reports from patients and clinicians. It holds 429 reports naming articaine, and the FDA flagged 63% of those reports as serious. The effects reported most often — leaving out reports about overdose, misuse or the condition being treated, which dominate the raw list for common medicines:
- dyspnoea54 reports
- hypersensitivity31 reports
- hypertension31 reports
- nausea31 reports
- pruritus31 reports
- anaphylactic reaction27 reports
- loss of consciousness25 reports
- tachycardia25 reports
Read these as a signal, not a rate. A report does not mean articaine caused the effect — anyone can file one, and many describe people taking several medicines for several conditions. Crucially there is no denominator: FAERS does not record how many people took the drug, so these counts cannot be turned into “X% of patients” — a bigger number often just means a more widely used or more talked-about drug. Duplicates exist, and publicity drives reporting. For what is actually established, read the FDA label section above.
Source: openFDA drug/event (FAERS), retrieved July 25, 2026.
Related calculators
Frequently asked questions
Can you take articaine with other medicines?
It depends on the medicine. We check it against the FDA labels rather than guessing: our interaction checker searches each drug's own label for the other and quotes what it says, naming the section it came from. Run articaine against whatever else you take — and remember that a label not naming a drug is not the same as that combination being safe.
What forms does articaine come in?
Across the brands we track, articaine is currently marketed as drops, per the FDA's National Drug Code Directory. Each form is dosed differently — follow the label for the exact product you were prescribed.
Is there a generic articaine?
We do not currently list a generic-labelled articaine product. That does not always mean none exists — it means none appears under a generic name in the FDA data we track. Ask your pharmacist.
Cite this page
- APA
- pharmaranks. (2026, July 24). Articaine: uses, dosing, side effects & brands. https://pharmaranks.com/drugs/articaine
- MLA
- “Articaine: uses, dosing, side effects & brands.” pharmaranks, 24 July 2026, https://pharmaranks.com/drugs/articaine.
We summarise public FDA and NIH sources — for a clinical claim, cite the primary source we link to as well.
Sources: FDA openFDA drug label, National Drug Code Directory, and Enforcement (recall) database. This page reproduces public FDA data and is not medical advice. Dosing is set by your prescriber.
Read the full FDA label for articaine on DailyMed (NIH) ↗.